Trelagliptin Succinate SYR-472 100mg Safety Evaluation of Powder CAS 1029877-94-8 CAS NO.1029877-94-8

Min.Order: 100 Gram
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Keywords

1029877-94-8
Trelagliptin Succinate
SYR-472

Quick Details

ProName: Trelagliptin Succinate SYR-472 100mg S...
CasNo: 1029877-94-8
Molecular Formula: C18H20FN5O2.C4H6O4
Appearance: white crystalline powder
Application: Trelagliptin succinate is an antidiabe...
DeliveryTime: 2-4 days after confirming your payment...
PackAge: 100g/ bag, 2 kg/ bag, 25kg/ carton or ...
Port: Wuhan
ProductionCapacity: 20000 Kilogram/Day
Purity: 99%
Storage: Store in sealed containers at cool & d...
Transportation: By DHL, TNT, FedEx, HKEMS, UPS, Etc
LimitNum: 100 Gram

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Trelagliptin Succinate SYR-472 100mg Safety Evaluation of Powder CAS 1029877-94-8

Quick Detail:

SYR-472 is a novel once-weekly oral DPP-4 inhibitor for type 2 diabetes, which could be a treatment option when clinicians seek to improve medication adherence by reducing the number of required administrations.

Product name	Trelagliptin succinate
CAS NO.	1029877-94-8
Synonyms	Trelagliptin succinate
Category	Pharmaceutical Raw Materials,Active Pharmaceutical Ingredients,Bulk Drugs,Fine Chemicals.
Purity	99% Trelagliptin succinate
Appearance	Trelagliptin succinate powder
Shelf life	2 years
Usage	Trelagliptin succinate is an antidiabetic drug. Trelagliptin succinate is used to improve glycemic control in people with type 2 diabetes
Storage	Trelagliptin succinate should be stored in a well-closed container at low temperature, keep away from moisture, heat and light.

Trelagliptin Succinate Usage:

Trelagliptin(SYR-472) is a long acting dipeptidyl peptidase-4 (DPP-4) inhibitor that is being developed for the treatment of type 2 diabetes (T2D).Trelagliptin succinate is an antidiabetic drug. Trelagliptin succinate is used to improve glycemic control in people with type 2 diabetes

Trelagliptin Succinate Application:

Trelagliptin Succinate (SYR-472), a novel dipeptidyl peptidase-4 inhibitor, shows sustained efficacy by once-weekly dosing in type 2 diabetes patients.

In this study, we characterized in vitro properties of trelagliptin, which exhibited approximately 4- and 12-fold more potent inhibition against human dipeptidyl peptidase-4 than alogliptin and sitagliptin, respectively, and >10,000-fold selectivity over related proteases including dipeptidyl peptidase-8 and dipeptidyl peptidase-9. Kinetic analysis revealed reversible, competitive and slow-binding inhibition of dipeptidyl peptidase-4 by trelagliptin (t1/2 for dissociation ≈ 30 minutes).

X-ray diffraction data indicated a non-covalent interaction between dipeptidyl peptidase and trelagliptin. Taken together, potent dipeptidyl peptidase inhibition may partially contribute to sustained efficacy of trelagliptin.

Trelagliptin Succinate COA

Item	Specification	Result
Appearance	Powder	Conforms
Color	White Powder or Crystal	Conforms
Mesh Size	100% through 80% mesh size	Conforms
Identification	Identical to R.S. sample	Conforms
Trelagliptin Succinate	99%	Conforms
Loss on Drying	≤5.0%	3.11%
Ash	≤5.0%	Conforms
Solvents Residue	Meet Eur.Ph6.0<5.4>	Conforms
Pesticides Residue	Meet USP32<561>	Conforms
Lead(Pb)	≤3.0mg/kg	2.45
Arsenic(As)	≤2.0mg/kg	1.29
Cadmium(Cd)	≤1.0mg/kg	0.68
Mercury(Hg)	≤0.1mg/kg	0.07

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Hubei XinRunde Chemical Co., Ltd is a renowned pharmaceutical manufacturer. We can offer high quality products at competitive price in quick delivery with 100% custom pass guaranteed. Never stop striving to offer our best service is our philosophy. We have Flexible and Untraceable payment terms. As a leading manufacture, our products have been exported to Germany, Norway, Poland, Finland, Spain, UK, France, Russia, USA, Brazil, Mexico, Australia, Japan, Korea, Thailand, Indonesia, Uruguay and many other countries.

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Trelagliptin Succinate (SYR-472) 100mg Safety Evaluation of Powder CAS 1029877-94-8